/ Home
/ SUBMISSION

/ The BJOC
/ Diamond Open Access
/ Journal Statistics
/ Editorial Board
/ Community
/ Call for papers

/ Latest Articles
/ Most accessed
/ Thematic issues
/ Volumes
/ Authors

/ Alerts

/ TWITTER
/ LINKEDIN
/ Mastodon
/ RSS FEED

Empty search

Article Type

Publication Date Range

Search Tips

This search combines search strings from the content search (i.e. "Full Text", "Author", "Title", "Abstract", or "Keywords") with "Article Type" and "Publication Date Range" using the AND operator.

Search Examples

aromatic	the word “aromatic”
aromatic aldehyde	the word “aromatic” OR “aldehyde”
+aromatic +aldehyde	both words “aromatic” AND “aldehyde”
+aromatic -aldehyde	the word “aromatic” but NOT “aldehyde”
“aromatic aldehyde”	the exact phrase “aromatic aldehyde”
benz*	words which begin with “benz”, such as “benzene” or “benzyl”
benz*yl	words that begin with “benz” and end with “yl”, such as “benzyl” or “benzoyl”
benzyl~	words that are close to the word “benzyl”, such as “benzoyl” (i.e., fuzzy search)

BROWSE
Latest Articles
Most accessed
thematic issues
volumes
authors

BROWSE

Latest Articles Most Accessed Thematic Issues Volumes Authors

Author

1 article(s) from Potter, Barry V L

Accessing simply-substituted 4-hydroxytetrahydroisoquinolines via Pomeranz–Fritsch–Bobbitt reaction with non-activated and moderately-activated systems

Marco Mottinelli,
Mathew P. Leese and
Barry V. L. Potter

Beilstein J. Org. Chem. 2017, 13, 1871–1878, doi:10.3762/bjoc.13.182

PDF

Graphical Abstract

Figure 1: Non-steroidal templates from estradiol.

Jump to Figure 1

Scheme 1: Pomeranz–Fritsch and Pomeranz–Fritsch–Bobbitt reactions. Conditions: (a) conc. H₂SO₄; (b) benzene, ...

Jump to Scheme 1

Scheme 2: Designed synthesis of THIQ. Conditions: (a) NaBH(OAc)₃, CHCl₃, rt; (b) 6 M HCl or 70% HClO₄ (see Table 1),...

Jump to Scheme 2

Scheme 3: Side reaction during the double alkylation of 7 and possible reaction mechanism for the formation o...

Jump to Scheme 3

Scheme 4: Competition between the formation of 5- and 7-substituted THIQs. Conditions: (a) 6 M HCl, rt.

Jump to Scheme 4

Scheme 5: Formation of the 4-hydroxy and 4-methoxy-THIQs. Conditions: (a) 6 M HCl or 70% HClO₄, rt (see Table 3).

Jump to Scheme 5

Scheme 6: Competition between the formation of THIQs 10a,o,p and indoles 16a,o,p. Conditions: (a) 70% HClO₄, ...

Jump to Scheme 6

Scheme 7: Competition between 6- and 7-membered ring formation. Conditions: (a) NaBH(OAc)₃, CHCl₃, rt; (b) 2,...

Jump to Scheme 7

Scheme 8: Competition between ring formation para- or meta- to an activating group. Conditions: (a) NaBH(OAc)₃...

Jump to Scheme 8

Album

Supp Info

Full Research Paper

Published 06 Sep 2017

Full text

Other Beilstein-Institut Open Science Activities

/ Help / Support & Contact / Alerts / Privacy Policy / Terms & Conditions / Impressum